Nootropics IDRA 21 for Children Intelligence Development

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Product: IDRA 21
CAS: 22503-72-6
MF: C8H9ClN2O2S
MW: 232.69
Storage Temp.: Store at RT
Appearance: white to off-white crystalline powder
Usage: IDRA-21 inhibits AMPA receptor desensitization and enhances cognition by a related mechanism. IDRA-21 is more able to cross the blood-brain barrier than Cyclothiazide.

ANALYTICAL ITEMS SPECIFICATION ANALYTICAL RESULTS
Appearance White to Off-White Powder White powder
Related substances A single impurity≤0.5% 0.14%
Total impurities≤1.0% 0.35%
Loss on drying ≤0.5% 0.08%
Assay >98% 99.0%
Conclusion Confirms to Enterprise Standard

Product: Mexidol
CAS: 127464-43-1
MF: C8H11NO.C4H6O4
MW: 255.268
Storage Temp.: Store at RT
Appearance: white to off-white crystalline powder
Usage: It is notable that Emoxypine has a biochemical structure that resembles Pyridoxine, a form of Vitamin B6. With this semblance, some benefits of Pyridoxine are sometimes attributed to Emoxypine. Such benefits include function for the central nervous system and brain, as well as its positive influence to red and white blood cells formation.

ANALYTICAL ITEMS SPECIFICATION ANALYTICAL RESULTS
Appearance White to Off-White Powder White powder
Related substances A single impurity≤0.5% 0.09%
Total impurities≤1.0% 0.24%
Loss on drying ≤0.5% 0.09%
Assay >98.5% 99.2%
Conclusion Confirms to Enterprise Standard

IDRA-21 is an ampakine drug and a benzothiadiazine derivative. IDRA-21 is a chiral molecule, with (+)-IDRA-21 being the active form.

 

IDRA-21 shows nootropic effects in animal studies, significantly improving learning and memory. It is around 10-30 times more potent than aniracetam in reversing cognitive deficits, and produces sustained effects lasting for up to 48 hours after a single dose.

The mechanism for this action is thought to be through promoting the induction of long-term potentiation between synapses in the brain.

IDRA-21 does not produce neurotoxicity under normal conditions, although it may worsen neuronal damage following global ischemia after stroke or seizures.

In comparison to the benzoylpiperidine derived ampakine drugs, IDRA-21 was more potent than CX-516, but less potent than CX-546.

Newer benzothiadiazide derivatives with greatly increased potency compared to IDRA-21 have been developed,but these have not been researched to the same extent, with the benzoylpiperidine and benzoylpyrrolidine CX-series of drugs being favoured for clinical development, most likely due to more favourable toxicity profiles at high doses.

whatsapp:+8617707569722
web: http://www.roidraw.com
email: lucy@wumeitech.com